
AP1189 acetate
CAS No. 959850-74-9
AP1189 acetate ( —— )
产品货号. M28790 CAS No. 959850-74-9
AP1189acetate 是黑皮质素 1 和黑皮质素 3 受体的偏向激动剂。
纯度: >98% (HPLC)






规格 | 价格/人民币 | 库存 | 数量 |
2MG | ¥786 | 有现货 |
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5MG | ¥1126 | 有现货 |
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10MG | ¥1839 | 有现货 |
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25MG | ¥3337 | 有现货 |
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50MG | ¥4965 | 有现货 |
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100MG | ¥7063 | 有现货 |
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200MG | 获取报价 | 有现货 |
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500MG | 获取报价 | 有现货 |
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1G | 获取报价 | 有现货 |
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生物学信息
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产品名称AP1189 acetate
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注意事项本公司产品仅用于科研实验,不得用于人体或动物的临床与诊断
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产品简述AP1189acetate 是黑皮质素 1 和黑皮质素 3 受体的偏向激动剂。
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产品描述AP1189 acetate is a biased agonist at melanocortin 1 and melanocortin 3 receptors.(In Vitro):Added to macrophage cultures, AP1189 reduced cytokine release, an effect reliant on both MC1 and MC3 as evident from the use of Mc1r(-/-) and Mc3r(-/-) macrophages. No melanogenesis was induced by AP1189 in B16-F10 melanocytes.(In Vivo):Oral AP1189 elicited anti-inflammatory actions in peritonitis and, upon administration at the peak of inflammation, accelerated the resolution phase by ~3-fold.
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体外实验——
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体内实验——
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同义词——
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通路GPCR/G Protein
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靶点Melanocortin Receptor
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受体calmodulin
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研究领域——
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适应症——
化学信息
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CAS Number959850-74-9
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分子量358.35
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分子式C16H18N6O4
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纯度>98% (HPLC)
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溶解度——
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SMILESO=[N+](C1=CC=CC=C1N2C(/C=C/C=N/NC(N)=N)=CC=C2)[O-].CC(O)=O
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化学全称——
运输与储存
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储存条件(-20℃)
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运输条件With Ice Pack
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稳定性≥ 2 years
参考文献
1.Noriko Koizumi, et al. Combined agent for cell therapy of corneal endothelial cell. US10959997B2
产品手册




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